Conference Agenda
Technical Programme of AsBIC9
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Session Overview |
Date: Sunday, 09/Dec/2018 | |
3:00pm - 4:00pm |
Registration Venue: Auditorium Collection of Registration Kit Foyer of Auditorium |
4:00pm - 5:00pm |
Opening Ceremony Venue: Auditorium Guest-of-Honour: Prof Barry Halliwell Chairman of Biomedical Research Council, A*STAR; Senior Advisor, Academic Appointments and Research Excellence, Office of the Senior Deputy President and Provost, Tan Chin Tuan Centennial Professor, National University of Singapore |
5:00pm - 6:00pm |
Plenary Lecture 1 Venue: Auditorium Chair: Han Vinh Huynh Chi-Ming CHE The University of Hong Kong, Hong Kong S.A.R. (China) Plenary ANTI-CANCER METAL MEDICINES WITH N-HETEROCYCLIC CARBENE LIGANDS |
6:00pm - 8:30pm |
Welcome Reception |
Date: Monday, 10/Dec/2018 | ||||
9:00am - 10:00am |
Plenary Lecture 2 Venue: Auditorium Chair: Giorgia Pastorin Thomas WARD University of Basel, Switzerland Plenary ARTIFICIAL METALLOENZYMES: CHALLENGES AND OPPORTUNITIES |
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10:00am - 10:15am |
Morning Tea Break |
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10:15am - 12:00pm |
Session A1 Venue: Lecture Theatre 50 Chair: Yangzhong Liu Keynote TARGETING STRATEGIES FOR METAL-BASED ANTICANCER AGENTS 10:45am - 11:05am Invited KINETICS AND SPECIATION OF THE DHARA REACTION AS A FUNCTION OF TEMPERATURE AND THE I/PT RATIOS 11:05am - 11:25am Invited MULTIACTION PLATINUM ANTICANCER COMPLEXES 11:25am - 11:45am Invited TOLYTERPYRIDINE METAL COMPLEXES AS RADIOSENSITIZERS FOR CANCER TREATMENT |
Session B1 Venue: Lecture Theatre 51 Chair: Way-Zen Lee Keynote BIOMIMETIC APPROACHES TO SELECTIVE CATALYTIC OXIDATIONS BY NONHEME IRON COMPLEXES 10:45am - 11:05am Invited ARTIFICIAL PHOTOSYNTHESIS BY HETEROGENEOUS CATALYSIS AND PHOTOREDOX C-C BOND CLEAVAGE 11:05am - 11:25am Invited PENTANUCLEAR IRON CATALYSTS FOR WATER OXIDATION 11:25am - 11:45am Invited JAHN–TELLER CONTROL OF CATALYTIC PROGRESSION IN BIOLOGICAL WATER OXIDATION 11:45am - 12:05pm Invited REACTIVITY OF RUTHENIUM(III) PTERIN COMPLEXES IN HYDROGEN ATOM TRANSFER |
Session C1 Venue: Lecture Theatre 52 Chair: Ho Yu Au-Yeung Keynote TEXAPHYRINS AS DRUG CANDIDATES: LIFE DEATH AND ATTEMPTS AT RESURRECTION 10:45am - 11:05am Invited MULTIFUNCTIONAL THERANOSTIC AGENTS FOR CANCER IMAGING AND THERAPY 11:05am - 11:25am Invited TWO-PHOTON FLUORESCENT PROBE FOR HYPOXIC CANCER STEM CELL BY RESPONDING TO THE ENDOGENOUS NITROREDUCTASE 11:25am - 11:45am Invited CHIRAL CYCLENS – A NEW PLATFORM FOR BIO-IMAGING AND BIOMEDICAL APPLICATIONS 11:45am - 12:00pm Oral PLATINIUM(II) COMPLEX AS TWO-PHOTON PHOSPHORESCENT BIOIMAGING AGENT |
Session D1 Venue: Lecture Theatre 53 Chair: Michael R. Reithofer Keynote ORGANOMETALLICS-BASED SERS REPORTERS 10:45am - 11:05am Invited NANOMEDICINE FOR IMPROVING CHEMORADIOTHRAPY, REAL-TIME EVALUATING DRUG EFFICACY, AND ENHANCING IMMUNOTHERAPY IN CANCER TREATMENT 11:05am - 11:25am Invited IMAGING THE ELEMENTAL SIGNATURES OF DISEASE: THE PAST, PRESENT AND FUTURE OF ATOMIC PATHOLOGY 11:25am - 11:40am Oral TARGETED NANOPARTICLES FOR CANCER THERAPY – QUANTIFICATION OF NANOPARTICLE UPTAKE ON A SINGLE CELL LEVEL USING SINGLE CELL INDUCTIVELY COUPLED PLASMA MASS SPECTROMETRY (SC-ICP-MS) 11:40am - 11:55am Oral A GRAPHENE NANOMESH-BASED FLEXIBLE FIELD-EFFECT TRANSISTOR DEVICE WITH HIGH SENSITIVITY FOR CANCER MONITORING |
12:00pm - 1:00pm |
Lunch |
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1:00pm - 2:45pm |
Session A2 Venue: Lecture Theatre 50 Chair: Maria Babak Invited GOLD-BASED ANTIBODY DRUG CONJUGATES AS POTENTIAL CHEMOTHERAPEUTICS FOR BREAST CANCER 1:20pm - 1:40pm Invited NOVEL STRUCTURAL MOTIFS IN THE DESIGN OF ORGANOMETALLIC ANTICANCER AGENTS: BIOMOLECULE INTERACTION AND IMPACT ON THE MODE OF ACTION 1:40pm - 2:00pm Invited METAL-ARENE COMPLEXES: ANTICANCER AND OTHER INTERESTING PROPERTIES 2:00pm - 2:15pm Oral DEVELOPMENT OF NOVEL METHODOLOGIES FOR THE SYNTHESIS OF RU(II)-ARENE ANTICANCER AGENTS 2:15pm - 2:30pm Oral SYNTHESIS AND EVALUATION OF BIOLOGICAL ACTIVITIES OF ORGANOMETALLIC CONJUGATES OF MONASTROL |
Session B2 Venue: Lecture Theatre 51 Chair: Tsai-Te Lu Keynote METAL-OXYGEN INTERMEDIATES IN DIOXYGEN ACTIVATION CHEMISTRY 1:30pm - 1:50pm Invited APPLICATION OF IMIDAZOLE-BASED CHELATING LIGANDS TO FUNCTIONAL SYNTHETIC COMPLEXES MIMICKING THE DIOXYGEN ACTIVATING NON-HEME IRON SPECIES 1:50pm - 2:10pm Invited NITRIC OXIDE DIOXYGENATION REACTION AND NITRITE REDUCTION BY IRON AND MANGANESE COMPLEXES HOUSING TAML FRAMEWORK 2:10pm - 2:30pm Invited UTILITY OF ANTHRACENE SCAFFOLD FOR MODELING OF THE [FE]-HYDROGENASE ACTIVE SITE 2:30pm - 2:50pm Invited ACTIVATIONS OF DIOXYGEN AND NITROGEN OXIDES: CORRELATIONS OF N-CONFUSED PORPHYRIN PLATFORMS WITH BIOLOGICAL ACTIVE POCKETS |
Session C2 Venue: Lecture Theatre 52 Chair: Jing Zhao Invited BIOMOLECULAR PROBES AND CELLULAR REAGENTS DERIVED FROM LUMINESCENT RHENIUM(I), RUTHENIUM(II), AND IRIDIUM(III) COMPLEXES 1:20pm - 1:40pm Invited SINGLET OXYGEN-RESPONSIVE MOLECULES FOR PHOTODELIVERY OF NEUROTRANSMITTERS 1:40pm - 2:00pm Invited DEVELOPMENT OF BORON DIPYRROMETHENE BASED QUENCHERS AS KEY COMPONENTS OF SMART FLUORESCENT PROBES AND PHOTOTHERAPEUTIC AGENTS 2:00pm - 2:20pm Invited DOPAMINE LUMINESCENT DETECTION IN BIOLOGICAL MATRIX BY A COPPER(II) COMPLEX 2:20pm - 2:35pm Oral A NEW BIFUNCTIONAL CHELATOR FOR BISMUTH AND LEAD RADIOPHARMACEUTICALS: A MACROCYCLIC LIGAND WITH SEMICARBAZONE PENDANT GROUPS |
Session D2 Venue: Lecture Theatre 53 Chair: Wai Yip Fan Keynote MOLECULAR DESIGN OF METAL COMPLEXES FOR TUMOR TARGETING 1:30pm - 1:50pm Invited DINUCLEAR PLATINUM-NUCLEOBASE COMPLEXES FOR PROTEIN RECOGNITION 1:50pm - 2:10pm Invited TRANSITION METAL COMPLEXES IN BIOMIMETIC AND CATALYTIC APPLICATIONS 2:10pm - 2:25pm Oral HYDROGEN PEROXIDE AS A BIOLOGICALLY-RELEVANT REDUCTANT AND HYDRIDE DONOR 2:25pm - 2:40pm Oral TRANSMETALATION WITH A TITANIUM(IV) COMPOUND TRANSFORMS BIOFUNCTIONAL COPPER INTO A CYTOTOXIC AGENT |
2:45pm - 4:15pm |
AsBIC Steering Committee Meeting Venue: Seminar Room 1 Chair: Hongzhe Sun |
Poster Session 1 & Tea Break Venue: Foyer of Auditorium Poster THE THERMODYNAMIC AND KINETIC DESCRIPTION OF THE REACTIONS IN SOLUTIONS WITH CONSTANT PH Poster BENZIMIDAZOLIUM-DERIVED N-HETEROCYCLIC CARBENES BRIDGING THE GAP BETWEEN PEPTIDES AND METAL COMPLEXES Poster “ON WATER” ONE-POT GREEN SYNTHESIS, DFT STUDIES AND REACTIVITY TOWARDS DNA AND PROTEIN BSA OF NOVEL RU(II)-P-CYMENE-2-ARYL BENZIMIDAZOLE (BIZ), BENZOTHIAZOLE (BTZ) AND BENZOXAZOLE (BOZ) SCAFFOLDS: THE INFLUENCE OF REGIOISOMER ON CYTOTOXICITY Poster A NEW RU(II) COMPLEX: DNA/HSA-BINDING, ANTI-MIGRATION AND BIOLOGICAL PROPERTIES IN A HUMAN BREAST TUMOR CELL LINE Poster UNDERSTANDING THE MECHANISM-OF-ACTION OF PT(II)-BASED TYPE II ICD INDUCERS VIA PURPOSEFUL SCAFFOLD MODIFICATION Poster ANTI-LEISHMANIAL ACTIVITY OF ALKYL GALLIUM QUINOLINOLATO COMPLEXES Poster METALLOCENYL EBSELEN COMPLEX AND ITS ACTIVITY ON THIOREDOXIN REDUCTASE Poster GROUP-VIII METALLOCYCLIC CARBAMOYL COMPLEXES AS STRUCTURAL MODELS OF THE [FE]-HYDROGENASE ACTIVE SITE Poster LC-TOF-MS ANALYSIS OF ORGANORUTHENIUM ANTICANCER COMPOUNDS IN BIOLOGICAL SAMPLES Poster MAKING ORGANORUTHENIUM COMPLEXES MORE HYDROPHILIC APPLIED NOVEL L-PHENYLALANINE-DERIVED ARENE LIGAND Poster SYNTHESIS, CHARACTERISAION, DNA BINDING INTERACTIONS, AND BIOLOGICAL ACTIVITY OF NICKEL SCHIFF BASE COMPLEXES. Poster BISMUTH(III) PHOSPHINATE 1D-COORDINATION POLYMERS AS ANTIBACTERIAL AGENTS Poster FLUORESCENT SENSORS FOR BIOLOGICAL METAL IONS Poster INVESTIGATION OF ELECTRON TRANSFER REACTION OF PQQ-DEPENDENT PYRANOSE DEHYDROGENASE FROM COPRINOPSIS CINEREA AND ITS AMINO ACID SUBSTITUTION MUTANTS ON ELECTRODES Poster NEW LIGANDS FOR RADIOCHEMISTRY USING METAL-TEMPLATED SYNTHESIS Poster THE EFFECTS OF LIGAND SUBSTITUTION ON THE ACTIVITY OF MONOFUNCTIONAL PLATINUM COMPLEXES Poster SYNTHESIS, IN VITRO CYTOTOXICITY AND ANTICANCER ACTIVITY OF SOME CU(II) COMPLEXES CONTAINING N2S (THIOLATE) AND N4S (DISULFIDE) CORES Poster FLUORESCENT ORGANOMETALLIC ANTICANCER AGENTS TO INVESTIGATE TUMOR CELL COMPARTMENT SELECTIVITY Poster TOWARDS METALLOSUPRAMOLECULAR CAGES FOR ANTICANCER DRUG DELIVERY Poster SIDE CHAIN SPECIFIC REACTIONS OF ORGANOMETALLIC COMPOUNDS TO LYSOZYME AND THE IMPACT ON THE PROTEIN Poster ARENE-RUTHENIUM(II) COMPLEXES AS LYSOSOME TARGETED PHOTOACTIVATED CHEMOTHERAPEUTIC AGENTS Poster NEAR-IR LUMINESCENT LANTHANIDE COMPLEXES OF DTPA–BISAMIDE USING 2-AMINOANTHRAQUINONE AS CHROMOPHORIC LIGAND: PHOTOPHYSICAL ASPECTS AND BIOLOGICAL APPLICATION Poster ENHANCED NEUROACTIVE AND NEUROPROTECTIVE ACTIVITIES IN NEURONAL CELLS USING ASSEMBLED IRON-TANNIC COMPLEXES AS AUTOPHAGY ENHANCER Poster DUAL DNA DAMAGE AND CELL APOPTOSIS INDUCED BY A NAPHTHALIMIDE PLATINUM(II) COMPLEX Poster COPPER(II) SELECTIVE CHELATORS ATTENUATE COPPER-OVERLOAD INDUCED OXIDATIVE STRESS Poster BODIPY-APPENDED OXIDOVANADIUM(IV) COMPLEXES OF CURCUMIN: AUGMENTED STABILITY OF THE ‘DRUG’ AND MITOCHONDRIA-TARGETED VISIBLE LIGHT PHOTOCYTOTOXICITY Poster VANADYL ACETYLACETONATE – AN INHIBITOR OF CLASSICAL UNFOLDED PROTEIN RESPONSE (UPR) TARGET GENE EXPRESSION SENSITISES CANCER CELLS TO ER-STRESS. Poster IMMUNOSTIMULATING EFFECTS OF PLATINUM-BASED COMPLEXES ON MACROPHAGES Poster A PHOTO-REDUCIBLE PRODRUG OF CISPLATIN Poster RUTHENIUM METALLOCOMPLEXES DESIGNED FOR IN SITU CELL LABELLING Poster CELL CYCLE–DEPENDENT UPTAKE AND CYTOTOXICITY OF ARSENIC-BASED DRUGS IN SINGLE LEUKEMIA CELLS Poster VISCOSITY-SENSITIVE PLATINUM(II) SCHIFF BASE COMPLEXS FOR LUMINESCENCE IMAGING AND PHOTODYNAMIC THERAPY Poster DEVELOPMENT OF AMINOALKYL TRISCYCLOMETALATED IRIDIUM COMPLEXES FOR CELL IMAGING THROUGH STRUCTURAL MODIFICATION Poster METAL COMPLEXES AS SELECTIVE FLUORESCENT STAINS FOR EXTRACELLULAR VESICLES Poster PLATINUM(IV) PRODRUGS WITH DNA-REPAIR PROTEIN IN BRCA-PROFICIENT CANCER CELLS AS MAJOR TARGET Poster PT(IV) PRODRUG INHIBIT NUCLEOTIDE EXCISION REPAIR PATHWAY TO CIRCUMVENT CISPLATIN RESISTANCE Poster A MULTIFACETED STUDY OF RU(II) ARENE ANTICANCER DRUGS: MECHANISMS OF ACTION, BIOLOGICAL TARGETS AND IMMUNOGENICITY Poster DEVELOPMENT OF ANTICANCER RUTHENIUM (II) ARENE SULFIDOCARBOXYLATO COMPLEXES Poster CROSSLINKING ALLOSTERIC SITES ON THE NUCLEOSOME CORE PARTICLE Poster IS BISMUTH REALLY THE ‘GREEN’ METAL? EXPLORING THE ANTIMICROBIAL ACTIVITY AND CYTOTOXICITY OF ORGANO-BISMUTH COMPOUNDS Poster CROSS-LINKING ALLOSTERIC INTER-HISTONE SITES IN THE NUCLEOSOME WITH HETERO-BINUCLEAR METALLOAGENTS Poster DESIGN AND SYNTHESIS OF CISPLATIN ANALOGUES Poster DESIGN OF THERANOSTIC METAL COMPLEXES FOR MITOCHONDRIA-TARGETED AND CANCER-SPECIFIC THERAPY Poster NEW WATER-SOLUBLE COPPER(II) COMPLEXES WITH MORPHOLINE-THIOSEMICARBAZONE HYBRIDS: INSIGHTS INTO THE ANTICANCER AND ANTIBACTERIAL MODE OF ACTION Poster LIGHT-INDUCED DNA BREAK BY USING INVASION OF PNA WITH RU COMPLEX Poster SOLUTION STRUCTURES OF MONOMERIC AND HIGHER-ORDER HUMAN TELOMERIC G-QUADRUPLEX COMPLEXES INDUCED BY THE PLATINUM(II)-BASED TRIPOD Poster METAL-MEDIATE BASE PAIRS; THE MODIFICATION OF DNA FOR FUTURE NANO-ELECTRONICS Poster SENSING THE MICROPOLARITY OF ENDOPLASMIC RETICULUM WITH A COUMARIN/BODIPY-HYBRIDIZED RATIOMETIC PROBE Poster SENSING MANGANESE (II) Poster SEMICYANINE PROBES WITH DIFFERENT H2S TRACKING BEHAVIOR AND MITOCHONDRIA-TARGETING ABILITY IN MCF-7 CELLS Poster A THERMODYNAMICALLY STABLE SEVEN-COORDINATE, MONO(AQUATED) MANGANESE(II) COMPLEX AS T1-WEIGHTED MRI CONTRAST AGENT Poster TOWARDS THE MULTIMODAL ANALYSIS OF LYSOSOMAL REDOX STATES Poster PROBING INTRACELLULAR REDUCTION OF ANTICANCER PLATINUM(IV) PRODRUG COMPLEXES Poster A NEAR-INFRARED FLUORESCENT PROBE FOR AMYLOID-β AGGREGATES Poster A FRET-BASED FLUORESCENT PROBE FOR FE3+ IN AQUEOUS SOLUTION Poster METAL-CO ARE EFFICIENT MULTIMODAL PROBES FOR CLASSICAL FLUORESCENCE, IR-IMAGING, AND X-FLUORESCENCE IMAGING Poster A FRET-BASED RATIOMETRIC LABILE ZINC(II) SENSOR: 3D FLUORESCENT IMAGING, FLOW CYTOMETRIC TRACKING AND CISPLATIN-INDUCED ZINC(II) FLUCTUATION MONITORING Poster USING FLUORESCENT ARRAYS TO MONITOR ANALYTES IN BIOLOGICAL FLUIDS Poster FLUORESCENT COBALT BASED PROBES FOR STUDYING THE CELLULAR REDOX ENVIRONMENT Poster INTRACELLULAR OXYGEN CONCENTRATION IMAGING USING MESOPOROUS SILICA NANOPARTICLES MODIFIED PLATINUM-PORPHYRIN Poster UNDERSTANDING THE CHEMISTRY OF SILVER IN BIOLOGICAL ENVIRONMENTS AND THE DEVELOPMENT OF SILVER-CONTAINING MATERIALS FOR USE AS ANTIBACTERIAL AGENTS Poster HYDROGEN PEROXIDE ACTIVATABLE CHELATORS FOR ALLEVIATING COPPER(II) INDUCED CELLULAR TOXICITY Poster A SENSITIVE WATER-SOLUBLE REVERSIBLE OPTICAL PROBE FOR MERCURY (II) DETECTION Poster TUNING STRUCTURES AND PROPERTIES FOR DEVELOPING NOVEL CHEMICAL TOOLS TOWARD DISTINCT PATHOGENIC ELEMENTS IN ALZHEIMER’S DISEASE Poster STRUCTURAL BASIS FOR TRANSCRIPTIONAL REGULATION OF A NOVEL HEME SENSOR PROTEIN IN PATHOGENIC BACTERIA Poster PHOTO-STERILIZATION OF PSEUDOMONAS AERUGINOSA IN BIOFILM UTILIZING ITS HEME ACQUISITION SYSTEM Poster ENGINEERING FERRITIN NANOCAGE TO UNRAVEL ITS SELF-ASSEMBLY, IRON(II) ENTRY, TRANSIT AND EXIT Poster RELEASING IRON FROM FERRITIN PROTEIN NANOCAGE BY REDUCTIVE METHOD: THE ROLE OF ELECTRON TRANSFER MEDIATOR Poster CAN COPPER IONS MODULATE THE SELF-ASSEMBLY OF AMYLOID-Β? Poster HCBP1 PEPTIDE CONJUGATED RUTHENIUM COMPLEX FOR TARGETING HEPATOMA THERAPY Poster CONSTRUCTION OF RECEPTOR TYROSINE KINASE TARGETING FLUORESCENCE SENSOR AND BIOLOGICAL IMAGING |
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4:15pm - 5:15pm |
Plenary Lecture 3 Venue: Auditorium Chair: Fangwei Shao Hua ZHANG Nanyang Technological University, Singapore Plenary CRYSTAL PHASE-ENGINEERING OF NOVEL NANOMATERIALS |
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5:15pm - 6:30pm |
Session A3 Venue: Lecture Theatre 50 Chair: Diego Montagner Invited RUTHENIUM COMPLEXES AS MODULATOR OF METABOLISM AND IMMUNOTHERAPY IN GASTRIC CANCER 5:35pm - 5:50pm Oral INTRACELLULAR IRON DEPLETION BY NOVEL CU(II) MORPHOLINE-THIOSEMICARBAZONE HYBRIDS 5:50pm - 6:05pm Oral METALS IN MEDICINE: PHENOTYPIC CHANGES INDUCED IN BREAST CANCER CELLS TREATED WITH METAL COMPLEXES 6:05pm - 6:20pm Oral CAN FUSOBACTERIUM NUCLEATUM ADHESION PROTEINS INCREASE THE PROOXIDATIVE ACTIVITY OF METAL IONS? |
Session B3 Venue: Lecture Theatre 51 Chair: Tapan Kanti Paine Invited METAL COMPLEXES AS MITOCHONDRIA-TARGETING ANTICANCER AGENTS 5:35pm - 5:55pm Invited NEW T*PP LIPOPHILIC CATIONS FOR ENHANCED MITOCHONDRIAL UPTAKE 5:55pm - 6:15pm Invited EPIGENETIC MODULATION AND MULTIPLE TARGETING OF ANTICANCER METAL COMPLEXES 6:15pm - 6:30pm Oral TARGETING EPIGENETIC CHANGES: MULTITARGETED VORINOSTAT (SAHA)-DERIVED METAL COMPLEXES WITH POTENT ANTICANCER AND HISTONE DEACETYLASE INHIBITORY ACTIVITY |
Session C3 Venue: Lecture Theatre 52 Chair: Kien Voon Kong Invited TITANIA AND SILICA-BASED LIQUID MARBLES AND DRY LIQUIDS FOR ENVIRONMENTAL APPLICATIONS 5:35pm - 5:55pm Invited ELECTROCATALYSTS IMMOBILIZED WITHIN LIPOSOMES FOR ENERGY CONVERSION IN NEUTRAL AQUEOUS MEDIA 5:55pm - 6:10pm Oral PHOTOINDUCED METHANE HYDROXYLATION USING PHOTOSYSTEM II RECONSTITUTED MEMBRANES CONTAINING PARTICULATE METHANE MONOOXYGENASE 6:10pm - 6:30pm Invited LIGNOCELLULOSIC BIOMASS VALORIZATION THROUGH THE DEVELOPMENT OF NANOMATERIALS FOR VERSATILE APPLICATIONS |
Session D3 Venue: Lecture Theatre 53 Chair: Wei Xia Invited BIOLOGICAL INORGANIC CHEMISTRY FOR CANCER IMMUNOTHERAPY 5:35pm - 5:55pm Invited METAL AND METAL OXIDE NANOPARTICLES ACT AS SUPPLEMENTARY AGENTS THAT AFFECT GUT HOMEOSTASIS 5:55pm - 6:15pm Invited TAILORED LANTHANIDE-DOPED UPCONVERSION NANOMATERIALS FOR SENSING AND BIOAPPLICATIONS 6:15pm - 6:30pm Oral ATOMICALLY PRECISE HYBRID NANOPARTICLES WITH MULTIVALENT CAPABILITIES |
6:30pm - 8:30pm |
AsBIC Steering Committee Dinner |
Date: Tuesday, 11/Dec/2018 | ||||
9:00am - 10:00am |
Plenary Lecture 4 Venue: Auditorium Chair: Yaw Kai Yan Rui Kang TANG Zhejiang University, China Plenary MODIFICATION OF ORGANISMS BY INORGANIC MATERIALS |
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10:00am - 10:15am |
Morning Tea Break |
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10:15am - 12:00pm |
Session A4 Venue: Lecture Theatre 50 Chair: Janice Rae Aldrich-Wright Keynote PLATINUM ANTICANCER AGENTS; FROM MAGIC BULLETS TO CLUSTER BOMBS 10:45am - 11:05am Invited PLATINUM ANTICANCER DRUGS: THE MECHANISTIC STUDY AND NEW DRUG DESIGN 11:05am - 11:25am Invited FUNCTIONALIZATION AND DELIVERY OF PT(IV) ANTICANCER PRODRUGS 11:25am - 11:45am Invited TRANIPLATIN AND MONO-ETHACRAPLATIN: TWO RECENT EXAMPLES OF DUAL-ACTION PLATINUM(IV) ANTICANCER PRO-DRUGS 11:45am - 12:00pm Oral A PHOTOACTIVE PLATINUM(IV) ANTICANCER COMPLEX INHIBITS THIOREDOXIN-THIOREDOXIN REDUCTASE SYSTEM ACTIVITY BY INDUCED OXIDIZATION OF THE PROTEIN |
Session B4 Venue: Lecture Theatre 51 Chair: Loi H. Do Invited SYNTHETIC HEME THIOLATE AND HEME SELENOLATE FOR UNDERSTANDING CHEMISTRY OF CYTOCHROME P450 10:35am - 10:55am Invited REACTIVITY OF A VANADIUM-BOUND THIYL RADICAL: ACTIVATION OF O-H AND C-O BONDS IN WATER AND METHANOL 10:55am - 11:15am Invited ADVANCED EPR STUDIES OF METAL-OXO SPECIES 11:15am - 11:35am Invited FUNCTIONAL MONO- AND DI-NITROSYL DIIRON(II) COMPLEXES MEDIATE THE REDUCTION OF NO TO N2O WITH RELEVANCE FOR FLAVODIIRON NO REDUCTASES 11:35am - 11:50am Oral CONSTRUCTION OF ARTIFICIAL P450 PEROXYGENASE FOR CATALYTIC MONOOXYGENATION OF NON-NATIVE SUBSTRATES |
Session C4 Venue: Lecture Theatre 52 Chair: Ming-Hsi Chiang Keynote ACTIVATION OF CHEMO/IMMUNOTHERAPY IN TUMOR MICROENVIRONMENT 10:45am - 11:05am Invited BIOINORGANIC NANOPARTICLES FOR IN VIVO DIAGNOSIS AND THERAPY OF TUMOR METASTASIS 11:05am - 11:25am Invited TOWARDS WATER-SOLUBLE HISTIDIN-N-HETEROCYCLIC CARBENE STABILIZED OPTICALLY ACTIVE GOLD NANOPARTICLES 11:25am - 11:40am Oral PEPTIDE-STABILIZED PLATINUM NANOPARTICLES SELECTIVELY ATTACK LIVER CANCER CELLS 11:40am - 11:55am Oral DESIGN AND SYNTHESIS OF ENZYME RESPONSIVE NANOCARRIERS BASED ON MESOPOROUS SILICA NANOPARTICLES FOR TARGETED DRUG DELIVERY APPLICATIONS |
Session D4 Venue: Lecture Theatre 53 Chair: Guido H. Clever Keynote COMBINING NANOSCIENCE WITH METALLO-SUPRAMOLECULAR RECOGNITION OF DNA AND RNA TO ACHIEVE BIO-ACTIVITY 10:45am - 11:05am Invited PT(BPA)2+: A FLUOROGENIC PROBE FOR RNA QUADRUPLEX AND REAL TIME TRACKING OF TERRA RAN QUADRUPLEX IN LIVE CELLS 11:05am - 11:20am Oral BIOINORGANIC REDOX SWITCHES REGULATE ENZYMATIC ACTIVITIES OF DNA REPAIR PROTEINS 11:20am - 11:35am Oral THE MECHANISM OF EXCISION OF 8-OXO-G WITH THE HOGG1 BER ENZYME 11:35am - 11:50am Oral ANTITUMOR METAL COMPLEXES WITH 8-HYDROXYQUNINOLINE AND ITS DERIVATIVES |
12:00pm - 1:00pm |
Lunch |
Technical Workshop Venue: Seminar Room 1 Oral QUANTIFYING THE UPTAKE OF METAL BASED THERAPY DRUGS USING SINGLE CELL ICP-MS |
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1:00pm - 2:45pm |
Session A5 Venue: Lecture Theatre 50 Chair: Taotao Zou Keynote CHEMICAL TOOLS AND TACTICS TO STUDY MULTIPLE FACETS IN ALZHEIMER’S DISEASE 1:30pm - 1:50pm Invited THE THERAPEUTIC EFFECT OF ANTI-DIABETIC VANADYL COMPLEXES ON ALZHEIMER’S DISEASE 1:50pm - 2:10pm Invited ACTIVATION OF ANGIOGENESIS AND WOUND HEALING IN DIABETIC MICE USING NO-RELEASING DINITROSYL IRON COMPLEXES 2:10pm - 2:25pm Oral ANTI-ALZHEIMER’S DISEASE POTENTIAL OF METAL COMPLEXES |
Session B5 Venue: Lecture Theatre 51 Chair: Woon Ju Song Keynote CATCHING A GLIMPSE OF SUB-METALATED METALLOTHIONEIN SPECIES 1:30pm - 1:50pm Invited A STRUCTURAL PERSPECTIVE ON NICKEL DELIVERY TO UREASE 1:50pm - 2:10pm Invited THE MOLECULAR MECHANISM OF GALLIUM UPTAKE BY PSEUDOMONAS AERUGINOSA 2:10pm - 2:25pm Oral ZN(II) INDUCED METAL DETOXIFICATION AND ANTIBIOTIC RESISTANCE BY HISTIDINE KINASE CZCS IN PSEUDOMONAS AERUGINOSA 2:25pm - 2:40pm Oral INVESTIGATING THE MULTI-FUNCTIONAL ROLES OF BACTERIOFERRITIN FROM MYCOBACTERIUM TUBERCULOSIS |
Session C5 Venue: Lecture Theatre 52 Chair: Michèle Salmain Keynote CHIRAL RECOGNITION OF AGEING DISEASE RELATED G-QUADRUPLEX AND AMYLOID AGGREGATION 1:30pm - 1:50pm Invited THE DIVERSE ROLE OF MOLYBDENUM- AND TUNGSTEN-ENZYMES 1:50pm - 2:10pm Invited ARTIFICIAL METALLOPROTEINS CONSTRUCTED WITH PROTEIN ASSEMBLIES FOR BIONANO APPLICATIONS 2:10pm - 2:25pm Oral CUPIN PROTEINS AS VERSATILE MACROMOLECULAR LIGANDS 2:25pm - 2:45pm Invited THE RICH CHEMISTRY OF WEAK INTERACTION IN BLUE COPPER PROTEIN |
Session D5 Venue: Lecture Theatre 53 Chair: Han Vinh Huynh Keynote CRITICAL FACTORS IN DETERMINING THE REACTIVITY OF HYPOCHLORITE ADDUCTS OF METAL COMPLEXES 1:30pm - 1:50pm Invited MANGANESE-COMPLEXES AS SOD-MIMICS: FROM DESIGN TO EVALUATION IN CELLS: AN INORGANIC CELLULAR CHEMISTRY STORY… 1:50pm - 2:10pm Invited NONHEME MANGANESE(III)-SUPEROXO COMPLEXES: SYNTHESIS, CHARACTERIZATION AND REACTIVITY 2:10pm - 2:25pm Oral SYNTHETIC MODEL PLATFORMS WITH MNII SPIN-LABELS FOR NANOMETER-SCALE DISTANCES MEASUREMENTS BY HIGH-FIELD PULSE EPR |
2:45pm - 4:15pm |
Fruit Fest * 3:45 pm - Group Photo-Taking at Foyer of Auditorium * |
Poster Session 2 & Tea Break Venue: Foyer of Auditorium Poster REVEALING THE IMMUNE PERTURBATION OF BLACK PHOSPHORUS NANOMATERIALS TO MACROPHAGES BY UNDERSTANDING THE PROTEIN CORONA Poster HIGHLY POROUS BOVINE SERUM ALBUMIN HYDROGEL/BEADS FOR REMOVAL OF ORGANIC, INORGANIC AND BACTERIAL COMPONTENTS FROM WATER Poster AN INJECTABLE, SELF HEALING AND STRESS SUSTAINABLE HYDORGEL OF BSA AS FUNCTIONAL BIOCOMPATIBLE MATERIAL FOR CONTROLLED DRUG DELIVERY IN CANCER CELLS Poster COPPER PHOSPHATE MORINGA OLEIFERA COAGULANT PROTEIN (MOCP) HYBRID NANOFLOWERS FOR SELECTIVE DETECTION AND REMOVAL OF INORGANIC, TOXIC METAL IONS AND ORGANIC DYES FROM WATER Poster DEVELOPMENT OF BIODEGRADABLE NANOPHOTOSENSITIZERS: A DEVICE DESIGNED FOR PHOTODYNAMIC THERAPY APPLICATIONS Poster A DUAL-TARGETED MODULATOR OF Aβ AGGREGATION AND NEUROINFLAMMATION AGAINST ALZHEIMER'S DISEASE Poster NANOPARTICLE-BASED DELIVERY OF HUMAN PROTEASOMES FOR THE TREATMENT OF ALZHEIMER'S DISEASE Poster PREPARATION OF FLUORESCENT POLYMER DOT FROM THE CARBONIZED OF MNO2 NANOSHEETS ENCAPSULATED HYALURONIC ACID FOR SMART REDOX-RESPONSIVE RELEASE OF PACLITAXEL Poster IMMOBILIZATION OF TUNGSTEN CATALYST BY CATECHOL CHEMISTRY IN PROCESSING MICROREACTORS FOR EFFECTIVE KILLING OF BACTERIA BY NEAR-INFRARED LIGHT Poster BIOCOMPATIBLE HYALURONIC ACID-FUNCTIONALIZED TUNGSTEN OXIDE NANOPARTICLE FOR IN VITRO-IN VIVO TUMOR TARGETING AND NIR-ASSISTED PHOTOTHERMAL THERAPY Poster FLUORESCENT DETECTION OF MYCOBACTERIUM TUBERCULOSIS VIA A HYBRIDIZATION-BASED PULL-DOWN ASSAY USING SEMICONDUCTOR NANOPROBES Poster MATERIALS FOR IMPROVING EXTRACORPOREAL CARBON DIOXIDE REMOVAL EFFICIENCY Poster NATURE AND BIO-INSPIRED, CONJUGATED MATERIALS FOR HIGH PERFORMANCE PLASTIC ORGANIC ELECTRONICS Poster GADOLINIUM OXIDE-CONTAINING MINERALIZED NANOPARTICLES AS A CONTRAST AGENT FOR MULTIMODAL IMAGING Poster INTRACELLULAR NO-RELEASING MINERALIZED NANOPARTICLES FOR CANCER CHEMOTHERAPY Poster TRANSGLUTAMINASE MEDIATED PEGYLATION OF NANOBODIES FOR TARGETED NANO-DRUG DELIVERY Poster BIOSYNTHETIC AG2S NANOPARTICLES ARE BIOCOMPATIBLE PHOTOCATALYTIC CATALYST FOR THE DEGRADATION OF POLLUTANTS UNDER VISIBLE LIGHT Poster ANTIBACTERIAL BISMUTH BASED HYDROGELS Poster STRONTIUM-DOPED HYDROXYAPATITE NANOCARRIER SYSTEMS LOADED WITH MIR-34A FOR THE TREATMENT OF BONE METASTASIS OF BREAST CANCER THROUGH REGULATING BONE MICROENVIRONMENTS Poster VISIBLE LIGHT-INDUCED PHOTODELIVERY OF HYDROGEN SULFIDE (H2S) Poster ULTRABRIGHT LANTHANIDE NANOPARTICLES FOR BIOLABELLING Poster INVESTIGATING THE STRUCTURE AND METAL COORDINATION PATHWAY OF A PLANT METALLOTHIONEIN 2 PROTEIN FROM CICER ARIETINUM Poster PROBING THE INTERACTION OF ANTICANCER DRUG TEMSIROLIMUS WITH HUMAN SERUM ALBUMIN: MOLECULAR DOCKING AND SPECTROSCOPIC INSIGHT Poster DEVELOPMENT OF AN ARTIFICIAL CARBONIC ANHYDRASE WITH PROMISCUOUS FORMATE DEHYDROGENASE ACTIVITY Poster Α-OXIDATIVE DECARBOXYLATION REACTION OF FATTY ACID CATALYZED BY FATTY ACID SPECIFIC PEROXYGENASE Poster NECLU_MT1: IT IS A MATTER OF PROTONS Poster STEADY STATE KINETICS OF QUINOL OXIDATION BY NITRIC OXIDE REDUCTASE FROM NEISSERIA MENINGITIS Poster GROUP VIII METALLOENZYMES – A STUDY ON THE CONJUGATION PROCESS AND EFFECTS ON THE PROTEIN HOST Poster EVOLUTION OF DE NOVO METALLO-β-LACTAMASES BY TUNING INTERACTIONS BETWEEN SUBSTRATES AND MICROENVIRONMENTS Poster SCREENING OF N-SUBSTITUTED DIPEPTIDES IN SEARCH FOR NOVEL DECOY MOLECULES FOR THE BENZENE HYDROXYLATION CATALYZED BY CYTOCHROME P450BM3 Poster DIFFERENTIAL REACTIVITY OF METAL BINDING DOMAINS OF COPPER ATPASES TOWARDS CISPLATIN AND COLOCALIZATION OF COPPER AND PLATINUM Poster A NEW PATHWAY OF NITRITE REDUCTASE ENZYME ACTIVITY FOR NITRIC OXIDE PRODUCTION Poster FACTORS CONTROLLING EXPRESSION LEVELS OF PERIPLASMIC CU/ZN-SUPEROXIDE DISMUTASE IN ESCHERICHIA COLI Poster A MISFOLDING MECHANISM OF CU/ZN-SUPEROXIDE DISMUTASE UNDER OXIDATIVE CONDITIONS OF AMYOTROPHIC LATERAL SCLEROSIS Poster CONFORMATION-DEPENDENT TOXICITY OF CU/ZN-SUPEROXIDE DISMUTASE IN CAENORHABDITIS ELEGANS Poster A NETWORK FOR INTRACELLULAR COPPER DISTRIBUTION CONROLLED BY INTERACTIONS BETWEEN COPPER CHAPERONES Poster DIRECT OBSERVATION OF CATALYTIC REACTION OF NITRIC OXIDE REDUCTASE USING TIME-RESOLVED VIS/IR SPECTROSCOPY Poster PROSTHETIC GROUPS ASSOCIATION: IRON / ZINC PORPHYRIN AND OXO-MOLYBDENUM (DITHIOLENE) COMPLEX IN RELEVANCE TO SULFITE OXIDASE Poster A COMBIND ENZYME/MODEL STUDY OF THIOL DIOXYGENASES Poster TARGETING THE UNDRUGGABLE AND UNREACHABLE Poster COMPARING AND CONTRASTING THE DECOY MOLECULE SYSTEM WITH DIFFERENT MEMBERS OF THE CYP102 FAMILY Poster HEME-REGULATED MECHANISM OF TARGET SSDNA BINDING IN A REGULATOR, COLD SHOCK PROTEIN (CSP) Poster ENGINEERING FERRITIN PROTEIN NANOCAGE TO UNDERSTAND ITS SELF-ASSEMBLY AND SEPARATING ITS MODIFIED & HYBRID FORMS Poster RECONSITITUTION OF MANGANESE-SUBSTITUTED P450BM3 BY LIGATING HEME AND REDUCTASE DOMAINS WITH SORTASE A Poster BIOCHEMICAL PROPERTIES OF DOMAINS IN IRON-DEPENDENT ALCOHOL DEHYDROGENASE FROM THE HYPERTHERMOPHILIC ARCHAEON PYROCOCCUS HORIKOSHII OT3 Poster A STABLE 'END-ON' SUPEROXOCOPPER(II) COMPLEX Poster ENERGY-EFFICIENT HYDROGEN EVOLUTION BY FE−S ELECTROCATALYSTS: MECHANISTIC INVESTIGATIONS Poster CLICKABLE IRIDIUM CATALYST AS ANTICANCER METALLODRUGS Poster COPPER(II)-TETRAPEPTIDES MIMICKING THE ACTIVE SITE OF LACCASE AS CATALYST IN THE SYNTHESIS OF PRO-MESALAMINE DRUG Poster A COMBINED EXPERIMENTAL AND COMPUTATIONAL STUDY ON IMINOSEMIQUINONE COORDINATED OXIDOVANADIUM(V) COMPLEX BY REDOX ACTIVE ONS LIGAND Poster ABIOLOGICAL CATALYSIS BY THERMOSTABLE CYTOCHROME P450 Poster BIOORTHOGONAL CATALYSIS IN LIVING CELLS Poster PROTONATION AND REDUCTION OF CARBONYL-RICH DIIRON COMPLEXES: INSIGHTS INTO THE ELECTROCATALYTIC MECHANISM OF HYDROGEN FORMATION Poster A SWITCH FROM MECHANISTIC COMPETITION MEDIATED BY A COORDINATION BETWEEN TEMPERATURE AND CONCENTRATION EFFECTS IN THE OXIDATION REACTION OF [FEII(N4PY/TPA)](OTF)2 Poster PHOSPHATASE-LIKE ACTIVITY OF A ZINC(II) COMPLEX BEARING BIS(THIOSEMICARBAZONE) LIGAND: BIOMIMETIC DEPHOSPHORYLATION PROCESS OF GLUCOSE-6-PHOSPHATE Poster A STABLE CO(III)-IODOSYLBENZENE ADDUCT AND EFFECTS OF REDOX-INACTIVE METAL ION ON ELECTRON TRANSFER PROPERTIES Poster DIRECT NITROSOATION OF CYS RESIDUES IN BIOMOLECULES THROUGH COBALT-NO COMPLEX Poster RHENIUM CARBONYL COMPLEXES WITH 2-PYRIDYL-1,2,3-TRIAZOLE DERIVED LIGANDS: APPLICATIONS IN CATALYSIS AND PHOTOPHYSICAL STUDIES Poster NONHEME MANGANESE(III) SUPEROXO MIMICS: SYNTHESIS, CHARACTERIZATION AND REACTIVITY Poster AN UNPRECEDENTED NONHEME COBALT(III)-PEROXYNITRITO COMPLEX WITH LONGEVITY AND ITS INSIGHT FOR CONVERSION TO NITRATE PRODUCT Poster REDOX-ACTIVE BEHAVIOR OF A PPP LIGAND WITH A COBALT CENTER Poster A NOVEL METAL-LIGAND COOPERATION EMPLOYING A P-P BOND AS A REDOX RESERVOIR AND AN ACTIVE REACTION SITE Poster CAFFEINE DEMETHYLATION BY THERMOPHILIC CYTOCHROMEP450 FROM SULFOLOBUS TOKODAII STRAIN 7 Poster THE EFFECT OF PHOSPHATE BUFFER ON THE FENTON REACTION-A DFT STUDY Poster INTERPLAY OF ELECTRONIC COOPERATIVITY AND EXCHANGE COUPLING IN REGULATING THE REACTIVITY OF DIIRON(IV)-OXO COMPLEXES TOWARDS C−H AND O−H BOND ACTIVATION Poster OXIDATION OF METHANE BY AN N-BRIDGED HIGH-VALENT DIIRON–OXO SPECIES: ELECTRONIC STRUCTURE IMPLICATIONS ON THE REACTIVITY Poster ANALYSIS OF FLUORIDE CONCENTRATION IN A CASCADE TANK SYSTEM IN ANURADHAPURA, SRI LANKA Poster PHOTOCHEMICAL REACTION OF AMINO ACID SCHIFF BASE METAL COMPLEX WITH HYDROXYL GROUP AND TITANIUM OXIDE COMPOSITE Poster ELECTRICAL ENERGY EXTRACTION IN THE PROCESS OF AN ENZYMATIC GALACTARIC ACID SYNTHESIS Poster SUPRAMOLECULAR METALLOGELS DERIVED FROM NUCLEOTIDE COORDINATION WITH INTRINSIC PEROXIDASE ACTIVITY FOR CONTROLLED RELEASE OF DRUG Poster PROGRESSIVE RELEASE OF MESOPOROUS NANO-SELENIUM DELIVERY SYSTEM FOR THE MULTI-CHANNEL SYNERGISTIC TREATMENT OF ALZHEIMER'S DISEASE |
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4:15pm - 5:15pm |
Plenary Lecture 5 Venue: Auditorium Chair: Han Sen Soo Abhishek DEY Indian Association for the Cultivation of Science, India Plenary BIO-INSPIRED ELECTROCATALYSTS |
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5:15pm - 6:30pm |
Session A6 Venue: Lecture Theatre 50 Chair: Christian Gaiddon Invited AURANOFIN INHIBITS VIRULENCE IN PSEUDOMONAS AERUGINOSA 5:35pm - 5:55pm Invited GOLD: NOT JUST JEWELRY… 5:55pm - 6:10pm Oral GOLD AND PLATINUM COMPLEXES CONTAINING N-HETEROCYCLIC CARBENE LIGANDS: ANTI-CACNER AGENTS AND LUMINESCENT BIOLOGICAL PROBES 6:10pm - 6:30pm Invited REDOX-ACTIVE GOLD(I) COMPLEXES AS DUAL TARGETING CANCER THERAPEUTIC AGENTS |
Session B6 Venue: Lecture Theatre 51 Chair: Jason England Invited CHARACTERIZATION OF SHORT-LIVED REACTION INTERMEDIATES OF NITRIC OXIDE REDUCASES BY TIME-RESOLVED TECHNIQUES 5:35pm - 5:55pm Invited NITRIC OXIDE DYNAMICS CONTROLLED BY FORMATION OF PROTEIN COMPLEX IN DENITRIFICATION 5:55pm - 6:10pm Oral LIGAND-METAL BOND IN CYTOCHROME C: INSIGHTS FROM STATIC AND TIME-DEPENDENT X-RAY SPECTROSCOPY 6:10pm - 6:30pm Invited SPECIFIC HEME BINDING IN IRON REGULATORY PROTEINS AND THEIR FUNCTIONAL SIGNIFICANCE |
Session C6 Venue: Lecture Theatre 52 Chair: Xiaogang Qu Invited THE TERMINAL ENZYME OF DENITRIFICATION 5:35pm - 5:55pm Invited HYDROXYLATION OF LINEAR ALKANES BY NON-HEME DI-IRON ALKANE HYDROXYLASE (ALKB) 5:55pm - 6:10pm Oral MYOGLOBIN RECONSTITUTED WITH MANGANESE PORPHYCENE FOR ARTIFICIAL METALLOENZYME CATALYZING C–H BOND HYDROXYLATION |
Session D6 Venue: Lecture Theatre 53 Chair: Felipe Garcia Invited ANTITUMOR METAL COMPLEXES BASED ON TRADITIONAL CHINESE MEDICINES ACTIVE INGREDIENT ALKALOIDS AND THEIR DERIVATIVES 5:35pm - 5:50pm Oral HALF-SANDWICH COMPLEXES OF QUINAZILIN-4-(3H)-ONE AS NEW ANTIPROLIFERATIVE ACTIVE AGENTS 5:50pm - 6:05pm Oral DEVELOPMENT OF BISMUTH THIOLATES AS POTENT BROAD-SPECTRUM INHIBITORS AGAINST B1 AND B2 METALLO-β-LACTAMASES 6:05pm - 6:20pm Oral DESIGN PRO-DRUG BASED ON THE LYS199 RESIDUE IN IIA SUB-DOMAIN OF HUMAN SERUM ALBUMIN |
6:30pm - 9:00pm |
Invited Speakers Dinner |
Young Researcher Networking Session |
Date: Wednesday, 12/Dec/2018 | |||
9:00am - 10:00am |
Plenary Lecture 6 Venue: Auditorium Chair: Bengang Xing Kazuya KIKUCHI Osaka University, Japan Plenary IN VIVO CHEMICAL PROBES FOR MRI AND FLUORESCENCE IMAGING |
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10:00am - 10:30am |
Graeme Hanson-AsBIC Early Career Researcher Award 2018 Venue: Auditorium Chair: Mi Hee Lim Award EMERGENCE AND EVOLUTION OF METALLOENZYMES |
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10:30am - 11:00am |
Morning Tea Break |
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11:00am - 1:00pm |
Session A7 Venue: Lecture Theatre 50 Chair: Shu-Sin Chng Keynote DISCOVERING NEW SIDEROPHORES THROUGH GENOME MINING 11:30am - 11:50am Invited BISMUTH COMPLEXES AS INHIBITORS AGAINST METALLO-BETA-LACTAMASE 11:50am - 12:10pm Invited METALLOCENE-CONTAINING COMPLEXES AS ANTIPARASITIC AND ANTIFUNGAL DRUG CANDIDATES 12:10pm - 12:25pm Oral CONJUGATION OF PLATINUM INTO MEFLOQUINE PROMOTES ANTIMALARIAL ACTIVITY AGAINST ASEXUAL STAGE 12:25pm - 12:40pm Oral DESIGN AND DEVELOPMENT OF ANTI-MICROBIAL BISMUTH-NANOCELLULOSE COMPOSITES |
Session B7 Venue: Lecture Theatre 51 Chair: Thomas Walczyk Invited STRUCTURE AND FUNCTION OF TRANSCRIPTIONAL REGULATOR ADOPTING HEME AS A SIGNALING MOLECLUE 11:20am - 11:35am Oral REGIONAL IRON DISTRIBUTION AND SOLUBLE FERROPROTEIN PROFILES IN THE HEALTHY HUMAN BRAIN 11:35am - 11:50am Oral STRUCTURAL BASIS FOR ENHANCEMENT OF HUMAN IRON UPTAKE BY DUODENAL FERRIC REDUCTASE WITH ASCORBATE 11:50am - 12:05pm Oral MECHANISTIC ASPECTS OF BIOLOGICAL CU(II) TRANSFERS 12:05pm - 12:20pm Oral METAL TOXICITY AND BIOAVAILABILITY IN SOIL AND WATER |
Session C7 Venue: Global Learning Room Chair: Youngmin You Keynote EBNA1-TARGETED INHIBITORS: THE NEW WAY FORWARD TO END EPSTEIN-BARR VIRUS ASSOCIATED CANCER 11:30am - 11:50am Invited LUMINESCENT LANTHANIDE PROBES AS TARGETED THERANOSTIC AND BIOIMAGING AGENTS 11:50am - 12:10pm Invited ULTRABRIGHT LANTHANIDE NANOPARTICLES FOR MICROSCOPY AND FLUOROIMMUNOLOGY 12:10pm - 12:30pm Invited DESIGN OF PERSISTENT LUMINESCENCE NANOPROBE FOR BIOMEDICAL APPLICATIONS 12:30pm - 12:50pm Invited STUDIES ON THE SMART LUMINESCENT MATERIALS BASED ON RARE EARTH COMPLEXES |
1:00pm - 2:00pm |
Lunch ~ 12:15 pm - 3:00 pm | Special luncheon for Plenary & Keynote Speakers (Ocean Restaurant, Resorts World Sentosa) ~ |
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2:00pm - 6:00pm |
Excursion |
Date: Thursday, 13/Dec/2018 | |||
9:00am - 10:00am |
Plenary Lecture 7 Venue: Auditorium Chair: John H Dawson Marcetta DARENSBOURG Texas A&M University, USA Plenary NITRIC OXIDE ASSISTED FIRST ROW TRANSITION METALS FOR HYDROGENASE-INSPIRED HER ELECTROCATALYSIS |
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10:00am - 10:30am |
Graeme Hanson-AsBIC Early Career Researcher Award 2018 Venue: Auditorium Chair: Christian Hartinger Award TRANSLATION OF BIOINSPIRED COORDINATION COMPLEXES & MATERIALS INTO BIOMEDICAL APPLICATIONS |
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10:30am - 11:00am |
Morning Tea Break |
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11:00am - 1:00pm |
Session A8 Venue: Lecture Theatre 50 Chair: Guangyu Zhu Keynote LANTHANIDES IN BIOLOGY AND MEDICINE 11:30am - 11:50am Invited IRIDIUM SIMCATS TO THE RESCUE 11:50am - 12:10pm Invited PHOTOPHYSICAL AND BIOLOGICAL ACTIVITY OF CYCLOMETALATED IRIDIUM(III) COMPLEX-PEPTIDE CONJUGATES SYNTHESIZED BY POST-COMPLEXATION FUNCTIONALIZATION 12:10pm - 12:25pm Oral BIOORTHOGONAL PHOTOACTIVATION OF METAL-BASED ANTICANCER PRODRUGS 12:25pm - 12:40pm Oral PHOTO-TRIGGERABLE TRACELESS STAUDINGER_BERTOZZI LIGATION REACTION: A VERSATILE PHOTO-CONTROLLABLE TOOL FOR PEPTIDE SYNTHESIS |
Session B8 Venue: Lecture Theatre 51 Chair: Weng Kee Leong Keynote ARTIFICIAL METALLOENZYMES DESIGN FOR ASYMMETRIC CATALYSIS IN AQUEOUS MEDIA 11:30am - 11:50am Invited ASSEMBLY AND ENZYMATIC FUNCTIONAL SIMULATION OF METAL-ORGANIC ARCHITECTURES 11:50am - 12:10pm Invited BIOCOMPATIBLE METAL CATALYSIS 12:10pm - 12:30pm Invited SELECTIVE CO2 CONVERSION AT A SINGLE NICKEL CENTER 12:30pm - 12:50pm Invited DEVELOPMENT OF USEFUL FUNCTIONAL MOLECULES BASED ON BIOINSPIRED COMPLEXES 12:50pm - 1:10pm Invited BIOORGANOMETALLIC B12 AS BIOINSPIRED CATALYST FOR GREEN ORGANIC SYNTHESIS |
Session C8 Venue: Global Learning Room Chair: Gilles Gasser Keynote CLICK FUNCTIONALIZATION OF PEPTIDES AND PROTEINS: NEW TOOLS FOR INORGANIC CHEMICAL BIOLOGY 11:30am - 11:50am Invited THE GROUP 13 METALLOSALENS IN BIOLOGICAL STUDIES 11:50am - 12:05pm Oral METAL-NTA-BASED FLUORESCENCE PROBES FOR LABELING PROTEINS INSIDE LIVING CELLS 12:05pm - 12:20pm Oral DUAL FLUOROPHORE HYBRIDIZATION: RATIOMETRIC SENSOR DESIGN AND CELL IMAGING 12:20pm - 12:40pm Invited FLUORESCENT DETECTION OF INTRACELLULAR CADMIUM ION BY CARBOHYDRATE-PENDANT POLYQUINOLINE LIGANDS 12:40pm - 12:55pm Oral AUTOFLUORESCENCE-FREE TARGETED TUMOR IMAGING BASED ON PERSISTENT LUMINESCENCE NANOPARTICLES |
1:00pm - 2:00pm |
Lunch |
SBIC Assembly Venue: Auditorium Chair: Sue Berners-Price |
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2:00pm - 4:00pm |
Session A9 Venue: Lecture Theatre 50 Chair: Fangwei Shao Keynote THE WORLD OF NON-CANONICAL NUCLEIC ACIDS 2:30pm - 2:50pm Invited FROM THEORETICAL CALCULATIONS TO SINGLE MOLECULES: A METAL-ION-DIRECTED SPLICE-SITE RNA-RNA INTERACTION 2:50pm - 3:10pm Invited TRANSITION METAL BINDING G-QUADRUPLEX DNA 3:10pm - 3:25pm Oral EFFICIENT HYDROLYTIC CLEAVAGE OF DNA AND ANTIPROLIFERATIVE EFFECT ON HUMAN CANCER CELLS BY COMPLEXES OF CU(II) AND ZN(II) 3:25pm - 3:40pm Oral SELECTIVE RECOGNITION OF DNA G-QUADRUPLEX AND I-MOTIF STRUCTURES BY A THIAZOLE ORANGE APPENDED CYCLEN IN THE PRESENCE OF CU(II) ION 3:40pm - 3:55pm Oral REDOX-CATALYZING DEOXYRIBOZYMES COMPOSED OF HEME AND DNAS |
Session B9 Venue: Lecture Theatre 51 Chair: Muhammad Hanif Invited MYOGLOBIN RECONSTITUTED WITH A CORRINOID METAL COMPLEX 2:20pm - 2:40pm Invited RATIONAL DESIGN OF FUNCTIONAL HEME ENZYMES IN MYOGLOBIN USING POST-TRANSLATIONAL MODIFICATIONS (PTMS) 2:40pm - 3:00pm Invited NEW INSIGHTS INTO TYROSINASE MECHANISM 3:00pm - 3:20pm Invited DEVELOPMENT OF RHENIUM CARBONYL-DRUG-PEPTIDE NANOPARTICLES FOR THERANOSTIC APPLICATIONS 3:20pm - 3:40pm Invited METAL-DEFICIENCY IN CU/ZN-SUPEROXIDE DISMUTASE: A POTENTIAL CAUSE OF MOTOR NEURON DISEASE, ALS 3:40pm - 4:00pm Keynote BIOMOLECULE/ORGANELLE-TARGETED ANTI-TUMOR METAL COMPLEXES |
Session C9 Venue: Global Learning Room Chair: Han Sen Soo Keynote TRANSITION METAL SIGNALING: BIOINORGANIC CHEMISTRY BEYOND ACTIVE SITES 2:30pm - 2:50pm Invited BIO-INSPIRED COPPER COMPLEXES FOR UNDERSTANDING THE CATALYTIC MECHANISM OF COPPER NITRITE REDUCTASE 2:50pm - 3:10pm Invited BIOINSPIRED DICOPPER COMPLEXES: CATALYTIC HYDROXYLATIONS OF INERT HYDROCARBONS WITH HYDROGEN PEROXIDE 3:10pm - 3:30pm Invited A STABLE END-ON (η1) SUPEROXOCOPPER(II) COMPLEX THAT DISPLAYS APPRECIABLE SUBSTRATE REACTIVITY 3:30pm - 3:50pm Keynote DINITROSYL IRON COMPLEXES (DNICS): SYNTHESIS TOWARD UNVEILING THE CATALYTIC ROLES OF DNICS |
4:00pm - 4:30pm |
Afternoon Tea Break |
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4:30pm - 5:30pm |
AsBIC Outstanding Achievement Award 2018 Venue: Auditorium Chair: Hongzhe Sun Award Lecture A JOURNEY FROM GOLD-BASED DRUG DESIGN TO METALLOGLYCOMICS Susan J. BERNERS-PRICE Griffith University, Australia |
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5:30pm - 6:30pm |
Prize Presentation, Closing & Handover Ceremony Venue: Auditorium |
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6:30pm - 7:00pm |
Proceed to Banquet |
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7:00pm - 11:00pm |
Banquet (ticketed event) |
Date: Friday, 14/Dec/2018 | |
9:00am - 12:00pm |
Visit to Nanyang Technological University Chair: Bengang Xing |
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